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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA PPP1R15B GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA ZC3H13 CTRPv2 pan-cancer AAC 0.21 4e-05
mRNA IKBIP GDSC1000 pan-cancer AAC 0.15 4e-05
mRNA TRPV5 CTRPv2 pan-cancer AAC 0.19 4e-05
mRNA DOLPP1 GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA PRUNE1 GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA HEYL GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA SETD1A GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA CACNG4 GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA PRDM7 GDSC1000 pan-cancer AAC 0.14 4e-05
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