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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA OAF CTRPv2 pan-cancer AAC 0.2 4e-05
mRNA TNS2 GDSC1000 pan-cancer AAC 0.14 4e-05
mRNA NTM GDSC1000 pan-cancer AAC 0.14 4e-05
mRNA UPF3B GDSC1000 pan-cancer AAC -0.13 4e-05
mRNA SOX5 CTRPv2 pan-cancer AAC 0.2 4e-05
mRNA DEFB134 CTRPv2 pan-cancer AAC 0.19 4e-05
mRNA POLR2F CTRPv2 pan-cancer AAC 0.21 4e-05
mRNA CMTM7 GDSC1000 pan-cancer AAC 0.13 4e-05
mRNA FGD3 GDSC1000 pan-cancer AAC -0.15 4e-05
mRNA HEY1 GDSC1000 pan-cancer AAC 0.13 4e-05
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