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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA PMP22 GDSC1000 pan-cancer AAC 0.15 3e-05
mRNA REC8 GDSC1000 pan-cancer AAC -0.13 3e-05
mRNA PARD3B GDSC1000 pan-cancer AAC -0.12 3e-05
mRNA ABLIM1 GDSC1000 pan-cancer AAC -0.14 3e-05
mRNA DYNLT3 CTRPv2 pan-cancer AAC 0.22 3e-05
mRNA PLA1A GDSC1000 pan-cancer AAC 0.14 3e-05
mRNA PI15 GDSC1000 pan-cancer AAC 0.14 3e-05
mRNA MPG CTRPv2 pan-cancer AAC 0.21 3e-05
mRNA ABCG5 GDSC1000 pan-cancer AAC 0.13 3e-05
mRNA WDR12 CTRPv2 pan-cancer AAC 0.21 3e-05
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