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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA TBC1D16 GDSC1000 pan-cancer AAC 0.22 8e-10
mRNA SPRY2 CTRPv2 pan-cancer AAC 0.31 9e-10
mRNA STRADB GDSC1000 pan-cancer AAC 0.19 9e-10
mRNA IL1RAPL1 GDSC1000 pan-cancer AAC 0.2 9e-10
mRNA HMCN1 CTRPv2 pan-cancer AAC 0.33 1e-09
mRNA EIF2AK4 GDSC1000 pan-cancer AAC 0.19 1e-09
mRNA LPL CTRPv2 pan-cancer AAC 0.27 1e-09
mRNA MBP GDSC1000 pan-cancer AAC 0.22 1e-09
mRNA TCP11 CTRPv2 pan-cancer AAC 0.27 1e-09
mRNA DNAH10 CTRPv2 pan-cancer AAC 0.29 1e-09
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