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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA DICER1 GDSC1000 pan-cancer AAC -0.12 9e-05
mRNA REM1 CTRPv2 pan-cancer AAC 0.18 9e-05
mRNA SLC26A4 GDSC1000 pan-cancer AAC 0.12 9e-05
mRNA AL137164.1 CTRPv2 pan-cancer AAC 0.18 9e-05
mRNA COLEC11 CTRPv2 pan-cancer AAC 0.19 9e-05
mRNA DNA2 GDSC1000 pan-cancer AAC -0.13 9e-05
mRNA HINFP GDSC1000 pan-cancer AAC -0.13 9e-05
mRNA ABCA9 CTRPv2 pan-cancer AAC 0.18 9e-05
mRNA PLEKHA6 GDSC1000 pan-cancer AAC -0.14 9e-05
mRNA MS4A7 CTRPv2 pan-cancer AAC 0.18 9e-05
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