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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA GEMIN2 GDSC1000 pan-cancer AAC -0.13 8e-05
mRNA ACSL6 CTRPv2 pan-cancer AAC 0.18 8e-05
mRNA SNTB1 CTRPv2 pan-cancer AAC 0.19 8e-05
mRNA PNPLA3 GDSC1000 pan-cancer AAC 0.14 8e-05
mRNA RNMT CTRPv2 pan-cancer AAC 0.2 8e-05
mRNA ATL2 GDSC1000 pan-cancer AAC -0.12 8e-05
mRNA TBX10 CTRPv2 pan-cancer AAC 0.19 8e-05
mRNA GLB1L CTRPv2 pan-cancer AAC 0.19 8e-05
mRNA LUZP6 CTRPv2 pan-cancer AAC 0.21 8e-05
mRNA PDIK1L GDSC1000 pan-cancer AAC -0.14 9e-05
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