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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA POLE3 GDSC1000 pan-cancer AAC -0.12 7e-05
mRNA MMP15 CTRPv2 pan-cancer AAC 0.2 7e-05
mRNA NPAS2 CTRPv2 pan-cancer AAC 0.19 7e-05
mRNA RFTN2 CTRPv2 pan-cancer AAC 0.2 7e-05
mRNA TMEM8A GDSC1000 pan-cancer AAC 0.12 7e-05
mRNA WDR35 GDSC1000 pan-cancer AAC 0.13 7e-05
mRNA DUSP26 GDSC1000 pan-cancer AAC -0.13 7e-05
mRNA SLC35B4 CTRPv2 pan-cancer AAC 0.23 7e-05
mRNA NAV3 CTRPv2 pan-cancer AAC 0.19 7e-05
mRNA HTN1 GDSC1000 pan-cancer AAC 0.12 7e-05
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