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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA LRCOL1 CTRPv2 pan-cancer AAC 0.31 4e-12
mRNA FAM167B GDSC1000 pan-cancer AAC 0.24 4e-12
mRNA SPRY2 GDSC1000 pan-cancer AAC 0.23 5e-12
mRNA ITIH6 CTRPv2 pan-cancer AAC 0.33 6e-12
mRNA L1TD1 CTRPv2 pan-cancer AAC 0.31 7e-12
mRNA PTCHD4 CTRPv2 pan-cancer AAC 0.34 8e-12
mRNA IFNGR2 CTRPv2 pan-cancer AAC 0.33 8e-12
mRNA VIP CTRPv2 pan-cancer AAC 0.32 9e-12
mRNA SPRED1 CTRPv2 pan-cancer AAC 0.36 1e-11
mRNA SH3TC2 CTRPv2 pan-cancer AAC 0.37 1e-11
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