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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
Dataset Select
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA FAM189A1 CTRPv2 pan-cancer AAC 0.33 4e-14
mRNA SPRED1 GDSC1000 pan-cancer AAC 0.25 5e-14
mRNA B4GALT6 CTRPv2 pan-cancer AAC 0.38 7e-14
mRNA GAS7 CTRPv2 pan-cancer AAC 0.41 1e-13
mRNA DKK4 CTRPv2 pan-cancer AAC 0.33 1e-13
mRNA MRGPRG CTRPv2 pan-cancer AAC 0.33 1e-13
mRNA ASCL5 CTRPv2 pan-cancer AAC 0.33 1e-13
mRNA LY6L CTRPv2 pan-cancer AAC 0.33 1e-13
mRNA CACHD1 CTRPv2 pan-cancer AAC 0.33 2e-13
mRNA GABRA1 CTRPv2 pan-cancer AAC 0.33 2e-13
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