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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA HTATSF1 GDSC1000 pan-cancer AAC -0.13 2e-05
mRNA PKM GDSC1000 pan-cancer AAC 0.13 2e-05
mRNA PODN CTRPv2 pan-cancer AAC -0.21 2e-05
mRNA SVIL CTRPv2 pan-cancer AAC 0.22 2e-05
mRNA GGT7 CTRPv2 pan-cancer AAC 0.22 2e-05
mRNA ITGA2 GDSC1000 pan-cancer AAC 0.16 2e-05
mRNA ASS1 GDSC1000 pan-cancer AAC -0.14 2e-05
mRNA FAM188B CTRPv2 pan-cancer AAC 0.2 2e-05
mRNA CSPG4 GDSC1000 pan-cancer AAC 0.16 2e-05
mRNA GRHL2 GDSC1000 pan-cancer AAC -0.16 2e-05
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