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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA ZFYVE16 GDSC1000 pan-cancer AAC 0.15 7e-06
mRNA MXRA7 GDSC1000 pan-cancer AAC 0.17 7e-06
mRNA CSGALNACT1 GDSC1000 pan-cancer AAC 0.14 7e-06
mRNA FAM129B GDSC1000 pan-cancer AAC 0.21 7e-06
mRNA STXBP1 CTRPv2 pan-cancer AAC 0.23 7e-06
mRNA BAG5 GDSC1000 pan-cancer AAC -0.14 7e-06
mRNA STK10 CTRPv2 pan-cancer AAC 0.27 7e-06
mRNA LLGL2 GDSC1000 pan-cancer AAC -0.18 7e-06
mRNA SYT17 GDSC1000 pan-cancer AAC -0.14 7e-06
mRNA TNFSF4 GDSC1000 pan-cancer AAC 0.14 7e-06
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