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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA NNMT GDSC1000 pan-cancer AAC 0.16 6e-06
mRNA GNS GDSC1000 pan-cancer AAC 0.15 6e-06
mRNA SHISA4 GDSC1000 pan-cancer AAC 0.17 6e-06
mRNA CAMSAP3 GDSC1000 pan-cancer AAC -0.17 6e-06
mRNA TXK CTRPv2 pan-cancer AAC 0.22 6e-06
mRNA ATM GDSC1000 pan-cancer AAC 0.16 6e-06
mRNA ZNF646 GDSC1000 pan-cancer AAC -0.15 7e-06
mRNA KLF13 GDSC1000 pan-cancer AAC -0.15 7e-06
mRNA MPV17 GDSC1000 pan-cancer AAC 0.14 7e-06
mRNA GYPC GDSC1000 pan-cancer AAC 0.2 7e-06
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