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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
Dataset Select
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA MOSPD2 CTRPv2 pan-cancer AAC 0.24 5e-06
mRNA MITF CTRPv2 pan-cancer AAC 0.25 5e-06
mRNA CAMK1D GDSC1000 pan-cancer AAC -0.15 5e-06
mRNA AP1S1 GDSC1000 pan-cancer AAC 0.15 5e-06
mRNA CXCL1 GDSC1000 pan-cancer AAC 0.15 5e-06
mRNA GJA3 CTRPv2 pan-cancer AAC 0.21 5e-06
mRNA TRIM26 GDSC1000 pan-cancer AAC -0.15 5e-06
mRNA AEN CTRPv2 pan-cancer AAC 0.22 5e-06
mRNA TYRP1 GDSC1000 pan-cancer AAC 0.16 5e-06
mRNA ACTN1 GDSC1000 pan-cancer AAC 0.17 5e-06
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