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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF106 CTRPv2 pan-cancer AAC 0.24 4e-06
mRNA POLR3G CTRPv2 pan-cancer AAC 0.23 4e-06
mRNA MAD2L1BP CTRPv2 pan-cancer AAC 0.23 4e-06
mRNA AP005242.1 CTRPv2 pan-cancer AAC 0.21 4e-06
mRNA CTHRC1 GDSC1000 pan-cancer AAC 0.15 4e-06
mRNA SLC24A1 GDSC1000 pan-cancer AAC 0.14 4e-06
mRNA RAB7B CTRPv2 pan-cancer AAC 0.24 4e-06
mRNA FAM167B CTRPv2 pan-cancer AAC 0.24 4e-06
mRNA CACHD1 GDSC1000 pan-cancer AAC 0.15 4e-06
mRNA PMP22 CTRPv2 pan-cancer AAC 0.26 4e-06
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