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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
Dataset Select
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA GPNMB CTRPv2 pan-cancer AAC 0.27 3e-06
mRNA OR5M1 GDSC1000 pan-cancer AAC -0.14 3e-06
mRNA ARHGAP33 GDSC1000 pan-cancer AAC -0.14 3e-06
mRNA CATIP GDSC1000 pan-cancer AAC -0.15 3e-06
mRNA DCAF12L2 GDSC1000 pan-cancer AAC -0.14 3e-06
mRNA SERPIND1 GDSC1000 pan-cancer AAC 0.14 4e-06
mRNA DPY19L1 GDSC1000 pan-cancer AAC 0.15 4e-06
mRNA SCARB1 GDSC1000 pan-cancer AAC 0.15 4e-06
mRNA SNAI2 GDSC1000 pan-cancer AAC 0.18 4e-06
mRNA ZNF711 GDSC1000 pan-cancer AAC -0.15 4e-06
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