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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA GSN GDSC1000 pan-cancer AAC 0.18 9e-07
mRNA AMER1 GDSC1000 pan-cancer AAC -0.16 1e-06
mRNA ATOX1 GDSC1000 pan-cancer AAC 0.16 1e-06
mRNA PCDHGA5 CTRPv2 pan-cancer AAC 0.28 1e-06
mRNA PCDHGB3 CTRPv2 pan-cancer AAC 0.28 1e-06
mRNA TMEM158 GDSC1000 pan-cancer AAC 0.17 1e-06
mRNA KIRREL CTRPv2 pan-cancer AAC 0.31 1e-06
mRNA NCK2 CTRPv2 pan-cancer AAC 0.25 1e-06
mRNA SHISA4 CTRPv2 pan-cancer AAC 0.28 1e-06
mRNA PCDHGA12 CTRPv2 pan-cancer AAC 0.28 1e-06
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