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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA ASPSCR1 CTRPv2 pan-cancer AAC 0.23 7e-07
mRNA SIRPA GDSC1000 pan-cancer AAC 0.18 7e-07
mRNA CRYL1 GDSC1000 pan-cancer AAC 0.16 8e-07
mRNA CD59 GDSC1000 pan-cancer AAC 0.17 8e-07
mRNA TMEM17 CTRPv2 pan-cancer AAC 0.26 8e-07
mRNA PCDHGA6 CTRPv2 pan-cancer AAC 0.28 8e-07
mRNA ZBTB5 GDSC1000 pan-cancer AAC -0.15 8e-07
mRNA HECA GDSC1000 pan-cancer AAC -0.16 8e-07
mRNA PPP1R27 CTRPv2 pan-cancer AAC 0.22 8e-07
mRNA STRBP GDSC1000 pan-cancer AAC -0.17 8e-07
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