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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA SHROOM2 CTRPv2 pan-cancer AAC 0.24 6e-07
mRNA PCDHGA3 CTRPv2 pan-cancer AAC 0.29 6e-07
mRNA LILRA5 CTRPv2 pan-cancer AAC 0.22 7e-07
mRNA ART3 CTRPv2 pan-cancer AAC 0.24 7e-07
mRNA CHCHD6 GDSC1000 pan-cancer AAC 0.17 7e-07
mRNA RETN CTRPv2 pan-cancer AAC 0.22 7e-07
mRNA STRA6 CTRPv2 pan-cancer AAC 0.23 7e-07
mRNA MELTF CTRPv2 pan-cancer AAC 0.26 7e-07
mRNA MYO10 GDSC1000 pan-cancer AAC 0.18 7e-07
mRNA CDH19 CTRPv2 pan-cancer AAC 0.27 7e-07
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