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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA DIS3L2 CTRPv2 pan-cancer AAC 0.23 4e-07
mRNA RBM8A GDSC1000 pan-cancer AAC -0.16 4e-07
mRNA NES CTRPv2 pan-cancer AAC 0.27 5e-07
mRNA GJB1 GDSC1000 pan-cancer AAC 0.17 5e-07
mRNA PTPN9 GDSC1000 pan-cancer AAC 0.15 5e-07
mRNA FABP7 CTRPv2 pan-cancer AAC 0.24 5e-07
mRNA KIF3C GDSC1000 pan-cancer AAC 0.17 5e-07
mRNA GLUD2 CTRPv2 pan-cancer AAC 0.25 5e-07
mRNA VDAC1 CTRPv2 pan-cancer AAC 0.23 5e-07
mRNA THEM4 GDSC1000 pan-cancer AAC 0.16 5e-07
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