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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA ACP5 CTRPv2 pan-cancer AAC 0.28 3e-07
mRNA ETV4 GDSC1000 pan-cancer AAC 0.18 3e-07
mRNA FGF1 CTRPv2 pan-cancer AAC 0.24 3e-07
mRNA PCDHGA11 CTRPv2 pan-cancer AAC 0.29 3e-07
mRNA DEFB136 CTRPv2 pan-cancer AAC 0.24 3e-07
mRNA SLC20A1 GDSC1000 pan-cancer AAC 0.16 3e-07
mRNA PAX3 GDSC1000 pan-cancer AAC 0.18 3e-07
mRNA TNFRSF14 GDSC1000 pan-cancer AAC 0.19 3e-07
mRNA MTFMT GDSC1000 pan-cancer AAC 0.15 4e-07
mRNA LAMA4 CTRPv2 pan-cancer AAC 0.27 4e-07
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