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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA C16orf52 CTRPv2 pan-cancer AAC 0.27 1e-07
mRNA LOXL3 CTRPv2 pan-cancer AAC 0.27 1e-07
mRNA PMEL GDSC1000 pan-cancer AAC 0.2 1e-07
mRNA FMN2 GDSC1000 pan-cancer AAC 0.17 1e-07
mRNA EMP3 GDSC1000 pan-cancer AAC 0.19 1e-07
mRNA ALDH1A3 CTRPv2 pan-cancer AAC 0.27 1e-07
mRNA IFT81 GDSC1000 pan-cancer AAC 0.18 1e-07
mRNA UCN2 CTRPv2 pan-cancer AAC 0.27 1e-07
mRNA RASGRF1 GDSC1000 pan-cancer AAC 0.16 1e-07
mRNA ELK3 GDSC1000 pan-cancer AAC 0.17 1e-07
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