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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA RPS27L GDSC1000 pan-cancer AAC 0.17 4e-08
mRNA MCAM CTRPv2 pan-cancer AAC 0.3 5e-08
mRNA LRRIQ3 GDSC1000 pan-cancer AAC 0.16 5e-08
mRNA PON2 GDSC1000 pan-cancer AAC 0.21 5e-08
mRNA HGFAC CTRPv2 pan-cancer AAC 0.25 5e-08
mRNA BIN3 GDSC1000 pan-cancer AAC 0.21 5e-08
mRNA RAB38 GDSC1000 pan-cancer AAC 0.19 5e-08
mRNA AATF CTRPv2 pan-cancer AAC 0.25 5e-08
mRNA CALML3 CTRPv2 pan-cancer AAC 0.25 5e-08
mRNA KIAA1755 CTRPv2 pan-cancer AAC 0.26 6e-08
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