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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA MSL2 GDSC1000 pan-cancer AAC -0.2 4e-08
mRNA PYGB CTRPv2 pan-cancer AAC 0.29 4e-08
mRNA KANK4 CTRPv2 pan-cancer AAC 0.25 4e-08
mRNA MCOLN3 CTRPv2 pan-cancer AAC 0.27 4e-08
mRNA VGF GDSC1000 pan-cancer AAC 0.18 4e-08
mRNA MYO5A CTRPv2 pan-cancer AAC 0.31 4e-08
mRNA TSR2 GDSC1000 pan-cancer AAC -0.16 4e-08
mRNA SEMA4C CTRPv2 pan-cancer AAC 0.26 4e-08
mRNA MPG GDSC1000 pan-cancer AAC 0.17 4e-08
mRNA PDGFA CTRPv2 pan-cancer AAC 0.26 4e-08
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