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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA SLC20A1 CTRPv2 pan-cancer AAC 0.26 3e-08
mRNA STK38 GDSC1000 pan-cancer AAC -0.17 3e-08
mRNA PTPRZ1 CTRPv2 pan-cancer AAC 0.26 3e-08
mRNA ISM1 CTRPv2 pan-cancer AAC 0.25 3e-08
mRNA MMP14 GDSC1000 pan-cancer AAC 0.21 3e-08
mRNA PRSS56 CTRPv2 pan-cancer AAC 0.25 3e-08
mRNA UPP1 GDSC1000 pan-cancer AAC 0.19 3e-08
mRNA ADGRB1 CTRPv2 pan-cancer AAC 0.25 3e-08
mRNA BACE2 GDSC1000 pan-cancer AAC 0.2 3e-08
mRNA NRP2 GDSC1000 pan-cancer AAC 0.18 3e-08
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