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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA GRIP2 CTRPv2 pan-cancer AAC 0.3 1e-11
mRNA C10orf90 GDSC1000 pan-cancer AAC 0.27 1e-11
mRNA SHC4 GDSC1000 pan-cancer AAC 0.25 2e-11
mRNA EXTL1 CTRPv2 pan-cancer AAC 0.34 2e-11
mRNA CTHRC1 CTRPv2 pan-cancer AAC 0.33 2e-11
mRNA ATP6V0E2 CTRPv2 pan-cancer AAC 0.33 2e-11
mRNA CYP17A1 CTRPv2 pan-cancer AAC 0.3 3e-11
mRNA SRPK3 CTRPv2 pan-cancer AAC 0.35 3e-11
mRNA APOC4-APOC2 CTRPv2 pan-cancer AAC 0.3 3e-11
mRNA ANKS1A CTRPv2 pan-cancer AAC 0.32 3e-11
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