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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA CLEC11A CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA LAMP5 CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA AMY2A CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA CCR6 CTRPv2 pan-cancer AAC 0.2 3e-09
mRNA SATB1 CTRPv2 pan-cancer AAC 0.21 3e-09
mRNA FRY CTRPv2 pan-cancer AAC 0.2 5e-09
mRNA AC243756.1 CTRPv2 pan-cancer AAC 0.19 7e-09
mRNA APOC4-APOC2 CTRPv2 pan-cancer AAC 0.2 8e-09
mRNA RP11-231C18.3 CTRPv2 pan-cancer AAC 0.19 1e-08
mRNA CLEC10A CTRPv2 pan-cancer AAC 0.19 1e-08
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