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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA AC025335.1 CTRPv2 pan-cancer AAC 0.086 0.02
mRNA AC073610.5 CTRPv2 pan-cancer AAC -0.073 0.03
mRNA AC084219.2 CTRPv2 pan-cancer AAC 0.093 0.009
mRNA AC087350.1 CTRPv2 pan-cancer AAC 0.092 0.01
mRNA AC090154.1 CTRPv2 pan-cancer AAC 0.082 0.03
mRNA AC104389.1 CTRPv2 pan-cancer AAC 0.13 0.0001
mRNA AC104389.2 CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA AC104534.3 CTRPv2 pan-cancer AAC 0.095 0.01
mRNA AC138969.4 CTRPv2 pan-cancer AAC 0.1 0.007
mRNA AC243756.1 CTRPv2 pan-cancer AAC 0.19 7e-09
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