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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA ZP1 CTRPv2 pan-cancer AAC 0.083 0.01
mRNA ZPBP CTRPv2 pan-cancer AAC -0.073 0.03
mRNA ZRANB3 CTRPv2 pan-cancer AAC 0.14 4e-05
mRNA ZSCAN12 CTRPv2 pan-cancer AAC 0.093 0.01
mRNA ZSCAN23 CTRPv2 pan-cancer AAC 0.12 0.003
mRNA ZSCAN4 CTRPv2 pan-cancer AAC 0.088 0.009
mRNA ZSCAN5A CTRPv2 pan-cancer AAC 0.1 0.004
mRNA ZSCAN9 CTRPv2 pan-cancer AAC 0.11 0.002
mRNA ZWINT CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA ZXDC CTRPv2 pan-cancer AAC 0.08 0.02
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