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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA PIM1 CTRPv2 pan-cancer AAC 0.26 2e-13
mRNA OR2B11 CTRPv2 pan-cancer AAC 0.25 2e-13
mRNA CFD CTRPv2 pan-cancer AAC 0.25 3e-13
mRNA GOLGA8O CTRPv2 pan-cancer AAC 0.25 4e-13
mRNA FLT3 CTRPv2 pan-cancer AAC 0.24 6e-13
mRNA GOLGA8Q CTRPv2 pan-cancer AAC 0.25 6e-13
mRNA NMUR1 CTRPv2 pan-cancer AAC 0.24 6e-13
mRNA GOLGA8K CTRPv2 pan-cancer AAC 0.24 1e-12
mRNA PLPPR3 CTRPv2 pan-cancer AAC 0.24 1e-12
mRNA LAIR1 CTRPv2 pan-cancer AAC 0.27 2e-12
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