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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA ZNF780B CTRPv2 pan-cancer AAC 0.094 0.008
mRNA ZNF784 CTRPv2 pan-cancer AAC 0.12 0.0004
mRNA ZNF8 CTRPv2 pan-cancer AAC 0.12 0.001
mRNA ZNF804B CTRPv2 pan-cancer AAC 0.089 0.007
mRNA ZNF808 CTRPv2 pan-cancer AAC 0.088 0.01
mRNA ZNF816 CTRPv2 pan-cancer AAC 0.082 0.02
mRNA ZNF816-ZNF321P CTRPv2 pan-cancer AAC 0.079 0.03
mRNA ZNF835 CTRPv2 pan-cancer AAC 0.077 0.03
mRNA ZNF865 CTRPv2 pan-cancer AAC 0.076 0.03
mRNA ZNF878 CTRPv2 pan-cancer AAC 0.099 0.006
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