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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA TYROBP CTRPv2 pan-cancer AAC 0.17 7e-07
mRNA KRTAP21-3 CTRPv2 pan-cancer AAC 0.17 7e-07
mRNA ZBTB3 CTRPv2 pan-cancer AAC 0.18 8e-07
mRNA PPIAL4C CTRPv2 pan-cancer AAC 0.16 9e-07
mRNA FRS3 CTRPv2 pan-cancer AAC 0.17 9e-07
mRNA IRF2BP2 CTRPv2 pan-cancer AAC 0.17 9e-07
mRNA TRERF1 CTRPv2 pan-cancer AAC 0.17 1e-06
mRNA LILRA1 CTRPv2 pan-cancer AAC 0.17 1e-06
mRNA EFCAB2 CTRPv2 pan-cancer AAC 0.17 1e-06
mRNA MTO1 CTRPv2 pan-cancer AAC 0.18 1e-06
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