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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA JUND CTRPv2 pan-cancer AAC 0.18 5e-08
mRNA RREB1 CTRPv2 pan-cancer AAC 0.19 5e-08
mRNA MYO1F CTRPv2 pan-cancer AAC 0.2 5e-08
mRNA PDGFRA CTRPv2 pan-cancer AAC 0.19 6e-08
mRNA HSD17B11 CTRPv2 pan-cancer AAC 0.2 7e-08
mRNA TOP1MT CTRPv2 pan-cancer AAC 0.2 7e-08
mRNA CTDP1 CTRPv2 pan-cancer AAC 0.21 7e-08
mRNA FAM45A CTRPv2 pan-cancer AAC 0.18 9e-08
mRNA ATP6V0A4 CTRPv2 pan-cancer AAC 0.18 1e-07
mRNA B3GNTL1 CTRPv2 pan-cancer AAC 0.18 1e-07
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