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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA PGC CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA VENTX CTRPv2 pan-cancer AAC 0.17 2e-07
mRNA FAM78A CTRPv2 pan-cancer AAC 0.24 2e-07
mRNA PDE7A CTRPv2 pan-cancer AAC 0.2 2e-07
mRNA CLASP2 CTRPv2 pan-cancer AAC 0.2 2e-07
mRNA SNX20 CTRPv2 pan-cancer AAC 0.22 3e-07
mRNA CD33 CTRPv2 pan-cancer AAC 0.19 3e-07
mRNA PHF7 CTRPv2 pan-cancer AAC 0.21 4e-07
mRNA STAR CTRPv2 pan-cancer AAC 0.18 5e-07
mRNA UTF1 CTRPv2 pan-cancer AAC 0.17 7e-07
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