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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA KCNN2 CTRPv2 pan-cancer AAC 0.23 1e-10
mRNA CISH CTRPv2 pan-cancer AAC 0.22 2e-10
mRNA CD300LF CTRPv2 pan-cancer AAC 0.22 4e-10
mRNA PARVG CTRPv2 pan-cancer AAC 0.24 7e-10
mRNA GOLGA8R CTRPv2 pan-cancer AAC 0.22 7e-10
mRNA MATK CTRPv2 pan-cancer AAC 0.22 9e-10
mRNA ZNF766 CTRPv2 pan-cancer AAC 0.22 1e-09
mRNA HRH4 CTRPv2 pan-cancer AAC 0.2 2e-09
mRNA APOC2 CTRPv2 pan-cancer AAC 0.2 3e-09
mRNA PPP1R27 CTRPv2 pan-cancer AAC 0.2 3e-09
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