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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA TARBP1 CTRPv2 pan-cancer AAC 0.17 4e-06
mRNA LINGO3 CTRPv2 pan-cancer AAC 0.17 4e-06
mRNA SSBP4 CTRPv2 pan-cancer AAC 0.16 5e-06
mRNA FRAT1 CTRPv2 pan-cancer AAC 0.17 5e-06
mRNA LRRC8C CTRPv2 pan-cancer AAC 0.16 6e-06
mRNA ADGRG5 CTRPv2 pan-cancer AAC 0.16 6e-06
mRNA NRROS CTRPv2 pan-cancer AAC 0.21 6e-06
mRNA PHF10 CTRPv2 pan-cancer AAC 0.16 6e-06
mRNA DOK2 CTRPv2 pan-cancer AAC 0.17 7e-06
mRNA AZU1 CTRPv2 pan-cancer AAC 0.15 8e-06
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