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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA SLC36A4 CTRPv2 pan-cancer AAC 0.078 0.03
mRNA CNKSR1 CTRPv2 pan-cancer AAC -0.092 0.03
mRNA ETV6 CTRPv2 pan-cancer AAC 0.079 0.03
mRNA PHC3 CTRPv2 pan-cancer AAC -0.073 0.03
mRNA GIT2 CTRPv2 pan-cancer AAC 0.093 0.03
mRNA C4B CTRPv2 pan-cancer AAC -0.073 0.03
mRNA AMBN CTRPv2 pan-cancer AAC 0.071 0.03
mRNA POLG2 CTRPv2 pan-cancer AAC 0.08 0.03
mRNA RAI14 CTRPv2 pan-cancer AAC -0.084 0.03
mRNA WDR6 CTRPv2 pan-cancer AAC 0.079 0.03
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