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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA SFMBT2 CTRPv2 pan-cancer AAC 0.08 0.03
mRNA NFKBIA CTRPv2 pan-cancer AAC -0.075 0.03
mRNA NLRP12 CTRPv2 pan-cancer AAC 0.072 0.03
mRNA CADM2 CTRPv2 pan-cancer AAC 0.075 0.03
mRNA SMPD3 CTRPv2 pan-cancer AAC 0.072 0.03
mRNA GPC1 CTRPv2 pan-cancer AAC -0.081 0.03
mRNA LARP7 CTRPv2 pan-cancer AAC 0.078 0.03
mRNA TRIM51 CTRPv2 pan-cancer AAC -0.083 0.03
mRNA DNAJC15 CTRPv2 pan-cancer AAC -0.075 0.03
mRNA SYNGAP1 CTRPv2 pan-cancer AAC 0.081 0.03
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