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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA AMY2B CTRPv2 pan-cancer AAC 0.18 1e-06
mRNA ACSM1 CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA LST1 CTRPv2 pan-cancer AAC 0.18 2e-06
mRNA PTPN7 CTRPv2 pan-cancer AAC 0.23 2e-06
mRNA LAIR2 CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA LMO2 CTRPv2 pan-cancer AAC 0.18 2e-06
mRNA ARHGAP45 CTRPv2 pan-cancer AAC 0.24 2e-06
mRNA TAF8 CTRPv2 pan-cancer AAC 0.16 2e-06
mRNA ZNF491 CTRPv2 pan-cancer AAC 0.17 2e-06
mRNA CTB-133G6.1 CTRPv2 pan-cancer AAC 0.2 2e-06
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