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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA IL17RA GDSC1000 pan-cancer AAC 0.1 0.004
mRNA NDC1 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA ZNF233 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA ATAD2 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA SAFB2 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA RP11-458D21.5 CTRPv2 pan-cancer AAC -0.1 0.004
mRNA TPM1 CTRPv2 pan-cancer AAC -0.13 0.004
mRNA CCDC71 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA RP11-701H24.9 CTRPv2 pan-cancer AAC 0.12 0.004
mRNA CHST2 CTRPv2 pan-cancer AAC 0.11 0.004
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