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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA CIB2 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA PRMT6 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA CBFA2T3 CTRPv2 pan-cancer AAC 0.12 0.004
mRNA FAM129B CTRPv2 pan-cancer AAC -0.12 0.004
mRNA PARP1 CTRPv2 pan-cancer AAC 0.12 0.004
mRNA MCM3 CTRPv2 pan-cancer AAC 0.12 0.004
mRNA RP11-468E2.1 CTRPv2 pan-cancer AAC -0.11 0.004
mRNA C7orf55-LUC7L2 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA RGPD1 CTRPv2 pan-cancer AAC 0.11 0.004
mRNA ATRN CTRPv2 pan-cancer AAC -0.12 0.004
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