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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA AGR3 CTRPv2 pan-cancer AAC -0.098 0.04
mRNA AC087651.2 CTRPv2 pan-cancer AAC 0.098 0.04
mRNA RP11-212D19.4 CTRPv2 pan-cancer AAC -0.096 0.04
mRNA EIF5AL1 CTRPv2 pan-cancer AAC -0.093 0.04
mRNA SREBF1 CTRPv2 pan-cancer AAC 0.095 0.04
mRNA STMN2 CTRPv2 pan-cancer AAC -0.12 0.04
mRNA MCM2 CTRPv2 pan-cancer AAC 0.11 0.04
mRNA ABCA5 CTRPv2 pan-cancer AAC 0.095 0.04
mRNA GCSAML CTRPv2 pan-cancer AAC -0.093 0.04
mRNA SYT17 CTRPv2 pan-cancer AAC 0.1 0.04
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