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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA MRPS22 CTRPv2 pan-cancer AAC -0.095 0.04
mRNA RGS4 CTRPv2 pan-cancer AAC -0.1 0.04
mRNA KIF3A CTRPv2 pan-cancer AAC 0.094 0.04
mRNA HIGD1C CTRPv2 pan-cancer AAC 0.095 0.04
mRNA SERPINB9 CTRPv2 pan-cancer AAC 0.097 0.04
mRNA STXBP5 CTRPv2 pan-cancer AAC -0.092 0.04
mRNA FIZ1 CTRPv2 pan-cancer AAC 0.096 0.04
mRNA ZNF589 CTRPv2 pan-cancer AAC 0.11 0.04
mRNA RP11-296A16.1 CTRPv2 pan-cancer AAC 0.096 0.04
mRNA STRBP CTRPv2 pan-cancer AAC 0.11 0.04
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