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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA RASSF1 CTRPv2 pan-cancer AAC -0.1 0.04
mRNA E2F3 CTRPv2 pan-cancer AAC 0.1 0.04
mRNA FAM227B CTRPv2 pan-cancer AAC -0.099 0.04
mRNA PSME4 CTRPv2 pan-cancer AAC 0.097 0.04
mRNA LDLRAD2 CTRPv2 pan-cancer AAC -0.1 0.04
mRNA SLFN14 CTRPv2 pan-cancer AAC -0.095 0.04
mRNA FZD2 CTRPv2 pan-cancer AAC 0.1 0.04
mRNA SLC38A10 CTRPv2 pan-cancer AAC 0.094 0.04
mRNA VARS CTRPv2 pan-cancer AAC 0.1 0.04
mRNA GYPB CTRPv2 pan-cancer AAC -0.093 0.04
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