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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA TRIM32 CTRPv2 pan-cancer AAC 0.13 0.007
mRNA CHD3 CTRPv2 pan-cancer AAC 0.13 0.007
mRNA U2AF1L4 CTRPv2 pan-cancer AAC 0.13 0.007
mRNA SH2B2 CTRPv2 pan-cancer AAC 0.14 0.007
mRNA UGGT1 CTRPv2 pan-cancer AAC 0.13 0.007
mRNA DAP CTRPv2 pan-cancer AAC -0.12 0.007
mRNA OPA3 CTRPv2 pan-cancer AAC 0.12 0.007
mRNA DHTKD1 CTRPv2 pan-cancer AAC 0.14 0.007
mRNA DDX39B CTRPv2 pan-cancer AAC 0.13 0.007
mRNA CROCC CTRPv2 pan-cancer AAC 0.12 0.007
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