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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA MYADML2 CTRPv2 pan-cancer AAC 0.13 0.004
mRNA EPM2A CTRPv2 pan-cancer AAC 0.14 0.004
mRNA PELI1 CTRPv2 pan-cancer AAC 0.14 0.004
mRNA WNT2B CTRPv2 pan-cancer AAC -0.13 0.004
mRNA ST6GAL1 CTRPv2 pan-cancer AAC 0.15 0.004
mRNA SLC31A1 CTRPv2 pan-cancer AAC -0.14 0.004
mRNA NFATC2 CTRPv2 pan-cancer AAC 0.16 0.004
mRNA ICA1 CTRPv2 pan-cancer AAC -0.15 0.004
mRNA OR4D1 CTRPv2 pan-cancer AAC -0.13 0.004
mRNA AC005042.1 CTRPv2 pan-cancer AAC -0.13 0.004
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