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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA RCVRN CTRPv2 pan-cancer AAC 0.14 0.002
mRNA STAT2 CTRPv2 pan-cancer AAC 0.15 0.002
mRNA FBXW12 CTRPv2 pan-cancer AAC 0.14 0.002
mRNA HNRNPUL1 CTRPv2 pan-cancer AAC 0.15 0.002
mRNA TAS2R13 CTRPv2 pan-cancer AAC -0.14 0.002
mRNA TP53AIP1 CTRPv2 pan-cancer AAC 0.14 0.002
mRNA GLTSCR1 CTRPv2 pan-cancer AAC 0.14 0.002
mRNA URGCP CTRPv2 pan-cancer AAC 0.15 0.002
mRNA ALOX5 CTRPv2 pan-cancer AAC 0.15 0.002
mRNA TRAF4 CTRPv2 pan-cancer AAC 0.15 0.002
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