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GSK1059615

Synonyms

SourcesNames Used
GRAY, CTRPv2GSK1059615
PharmacoGx GSK1059615

External IDs

DatabaseIdentifier
Smiles: C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4
Inchikey: QDITZBLZQQZVEE-YBEGLDIGSA-N
Pubchem: 23582824

Annotated Targets

PIK3CD, PIK3CG, MTOR, PIK3CA, PIK3CB

FDA Approval Status

Not Approved
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Top molecular features associated with response to GSK1059615


Feature TypeStandardized
Nominal ANOVA
mRNA LCN1 CTRPv2 pan-cancer AAC -0.093 0.03
mRNA WDR7 CTRPv2 pan-cancer AAC 0.11 0.03
mRNA PCDHGA11 CTRPv2 pan-cancer AAC 0.12 0.03
mRNA FAM188B CTRPv2 pan-cancer AAC 0.096 0.03
mRNA TGIF2 CTRPv2 pan-cancer AAC 0.11 0.03
mRNA DAZAP1 CTRPv2 pan-cancer AAC 0.12 0.03
mRNA LGALS7B CTRPv2 pan-cancer AAC -0.094 0.03
mRNA PCDHGB3 CTRPv2 pan-cancer AAC 0.12 0.03
mRNA RUNX1 CTRPv2 pan-cancer AAC -0.1 0.03
mRNA BICD2 CTRPv2 pan-cancer AAC 0.1 0.04
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