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GSK1120212

Synonyms

SourcesNames Used
GDSC1000Trametinib
GRAYGSK1120212
CTRPv2trametinib
PharmacoGx GSK1120212

External IDs

DatabaseIdentifier
Smiles: CC1=C2C(=C(N(C1=O)C)NC3=C(C=C(C=C3)I)F)C(=O)N(C(=O)N2C4=CC(=CC=C4)NC(=O)C)C5CC5
Inchikey: LIRYPHYGHXZJBZ-UHFFFAOYSA-N
Pubchem: 11707110

FDA Approval Status

Approved
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Top molecular features associated with response to GSK1120212


Feature TypeStandardized
Nominal ANOVA
mRNA KCNN4 CTRPv2 pan-cancer AAC 0.3 2e-09
mRNA PLXNB3 CTRPv2 pan-cancer AAC 0.3 4e-07
mRNA TRIB2 CTRPv2 pan-cancer AAC 0.3 1e-07
mRNA CST3 CTRPv2 pan-cancer AAC 0.29 1e-08
mRNA MMP17 CTRPv2 pan-cancer AAC 0.29 5e-07
mRNA ARHGEF11 CTRPv2 pan-cancer AAC 0.29 3e-07
mRNA PFKFB4 CTRPv2 pan-cancer AAC 0.29 2e-07
mRNA ARAP3 CTRPv2 pan-cancer AAC 0.29 2e-08
mRNA GSTK1 CTRPv2 pan-cancer AAC 0.29 8e-09
mRNA ADGRE5 CTRPv2 pan-cancer AAC 0.29 1e-08
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