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GSK1120212

Synonyms

SourcesNames Used
GDSC1000Trametinib
GRAYGSK1120212
CTRPv2trametinib
PharmacoGx GSK1120212

External IDs

DatabaseIdentifier
Smiles: CC1=C2C(=C(N(C1=O)C)NC3=C(C=C(C=C3)I)F)C(=O)N(C(=O)N2C4=CC(=CC=C4)NC(=O)C)C5CC5
Inchikey: LIRYPHYGHXZJBZ-UHFFFAOYSA-N
Pubchem: 11707110

FDA Approval Status

Approved
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Top molecular features associated with response to GSK1120212


Feature TypeStandardized
Nominal ANOVA
mRNA APBB1IP CTRPv2 pan-cancer AAC -0.27 3e-05
mRNA CPSF6 CTRPv2 pan-cancer AAC -0.27 4e-06
mRNA TAF5 CTRPv2 pan-cancer AAC -0.27 2e-06
mRNA SETD2 CTRPv2 pan-cancer AAC -0.27 2e-06
mRNA RP4-635E18.9 CTRPv2 pan-cancer AAC -0.27 9e-08
mRNA C14orf132 CTRPv2 pan-cancer AAC -0.27 2e-05
mRNA CKAP5 CTRPv2 pan-cancer AAC -0.27 7e-08
mRNA NUDT21 CTRPv2 pan-cancer AAC -0.26 2e-07
mRNA STRBP CTRPv2 pan-cancer AAC -0.26 1e-06
mRNA ZNF709 CTRPv2 pan-cancer AAC -0.26 4e-07
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