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GSK1120212

Synonyms

SourcesNames Used
GDSC1000Trametinib
GRAYGSK1120212
CTRPv2trametinib
PharmacoGx GSK1120212

External IDs

DatabaseIdentifier
Smiles: CC1=C2C(=C(N(C1=O)C)NC3=C(C=C(C=C3)I)F)C(=O)N(C(=O)N2C4=CC(=CC=C4)NC(=O)C)C5CC5
Inchikey: LIRYPHYGHXZJBZ-UHFFFAOYSA-N
Pubchem: 11707110

FDA Approval Status

Approved
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Top molecular features associated with response to GSK1120212


Feature TypeStandardized
Nominal ANOVA
mRNA MGST2 CTRPv2 pan-cancer AAC 0.25 3e-07
mRNA DUSP6 CTRPv2 pan-cancer AAC 0.25 3e-07
mRNA SLC20A1 CTRPv2 pan-cancer AAC 0.25 3e-07
mRNA PLXNB3 CTRPv2 pan-cancer AAC 0.3 4e-07
mRNA CD63 CTRPv2 pan-cancer AAC 0.3 4e-07
mRNA GPR35 CTRPv2 pan-cancer AAC 0.26 4e-07
mRNA C1orf162 CTRPv2 pan-cancer AAC 0.24 4e-07
mRNA ZNF709 CTRPv2 pan-cancer AAC -0.26 4e-07
mRNA LIN54 CTRPv2 pan-cancer AAC -0.25 4e-07
mRNA IFNGR2 CTRPv2 pan-cancer AAC 0.26 5e-07
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